Repozytorium

The analysis of the structural aspects of Cu(II) binding by cyclic His/Asp-analogues of somatostatin.

Autorzy

Aleksandra Marciniak

Aleksandra Kotynia

Marek Cebrat

Justyna Brasuń

Rok wydania

2020

Czasopismo

International Journal of Peptide Research and Therapeutics

Numer woluminu

26

Strony

969-977

DOI

10.1007/s10989-019-09900-9

Kolekcja

Naukowa

Język

Angielski

Typ publikacji

Artykuł

Streszczenie

Two new somatostatin analogs with a characteristic part of the sequence in their structures, -c(Cys-Phe-Trp-Lys-Thr-Cys)-, were synthesized and analyzed in terms of their coordination abilities with copper(II) ions. Cyclic peptides analyzed in our previous work had histidine and aspartic acid moieties in their structures which were responsible for metal ion coordination. In analyzed molecules these amino acids are also present. Peptides Ac[D1,2,9,10]c(SST) and Ac[H1,2,9,10]c(SST) have four aspartic acid or four histidine moieties, respectively. Both peptides bind Cu(II) effectively. Due to similar structures and the possibility of comparing the obtained results with these for the two previously published, the coordination abilities of two new ligands are possible to propose. Moreover, the effectiveness of copper(II) ion binding by four cyclic His/Asp-analogues of somatostatin is also discussed here. The peptide with four histidine moieties is the most efficient among described ligands.

Słowa kluczowe

Somatostatin, Somatostatin analogues, Copper complexes, Potentiometric measurements, Spectroscopy

Licencja otwartego dostępu

CC-BY

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Pełny tekst licencji: https://creativecommons.org/licenses/by/3.0/pl/legalcode

Adres publiczny

http://dx.doi.org/10.1007/s10989-019-09900-9

Strona internetowa wydawcy

http://link.springer.com

Podobne publikacje
2017

The coordination abilities of new cyclic analogs of somatostatin.

Marciniak Aleksandra, Cebrat Marek, Brasuń Justyna

2014

Structural aspects of copper(II) binding by a multi-His analogue of somatostatin.

Marciniak Aleksandra, Czyżnikowska Żaneta, Cebrat Marek, Kotynia Aleksandra, Brasuń Justyna