Repozytorium

Influence of solvent effect on polymorphism of 4-hydroxy-2-methyl-N-2-pyridyl-2H-1,2-benzothiazine-3-carboxamide-1,1-dioxide (piroxicam).

Autorzy

Maria Janik

Zbigniew Malarski

Jerzy Mroziński

Józef Wajcht

Zygmunt Zborucki

Rok wydania

1991

Czasopismo

Journal of Crystallographic and Spectroscopic Research

Numer woluminu

21

Strony

519-522

DOI

10.1007/BF01160669

Kolekcja

Naukowa

Język

Angielski

Typ publikacji

Artykuł

Streszczenie

Piroxicam (4-hydroxy-2-methyl-N-2-piridyl-2H- 1,2-benzothiazine-3-carboxamide- 1,1-dioxide), belongs to the class of acidic, nonsteroidal antiinflammatory (NSAI) drugs (Wiseman et al., 1976). Piroxicam is an effective analgesic agent in rheumatoid arthritis, anky- losing spondylitis, and acute pain in muskuloskeletal disorder and episiotomy. It can diminish or inhibit the development of all symptoms of inflammation no matter what its reason (Brogden et al., 1981). Piroxicam crys- tallizes in two modifications o~ and/3 (Fig. 1), in space groups Pca21 with Z = 4 and P21/c with Z = 4 (Reck et al., 1988; Kojir-Prodi6 and Ruzir-Toros, 1982), respectively. The conformation of the molecule in both structures is approximately planar and rigid, owing to the strong intramolecular hydrogen bonding O(17)--H...O(15) of lengths 2.526(2)A (cr and 2.561(5),~ (/3).

Słowa kluczowe

Physical chemistry, inorganic chemistry, Solvent effect, Piroxicam, organometallic chemistry

Adres publiczny

https://doi.org/10.1007/BF01160669

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