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Autor publikacji Justyna Piekielna-Ciesielska
Synthesis, Biological Activity and Molecular Docking of Chimeric Peptides Targeting Opioid and NOP Receptors
Wtorek Karol, Ghidini Alessia, Gentilucci Luca, Adamska-Bartłomiejczyk Anna, Piekielna-Ciesielska Justyna, Ruzza Chiara, Sturaro Chiara, Calò Girolamo, Pieretti Stefano, Kluczyk Alicja, McDonald John, Lambert David G., Janecka Anna
Synthesis, pharmacological evaluation, and computational studies of cyclic opioid peptidomimetics containing β3-lysine
Wtorek Karol, Lipiński Piotr F. J., Adamska-Bartłomiejczyk Anna, Piekielna-Ciesielska Justyna, Sukiennik Jarosław, Kluczyk Alicja, Janecka Anna
Pharmacological characterization of µ-opioid receptor agonists with biased G protein or β-arrestin signaling, and computational study of conformational changes during receptor activation.
Piekielna-Ciesielska Justyna, Artali Roberto, Azzam Ammar A. H., Lambert David G., Kluczyk Alicja, Gentilucci Luca, Janecka Anna
Design, synthesis and functional analysis of cyclic opioid peptides with Dmt-Tic pharmacophore.
Sarkar Arijit, Adamska-Bartłomiejczyk Anna, Piekielna-Ciesielska Justyna, Wtorek Karol, Kluczyk Alicja, Borics Attila, Janecka Anna
Pharmacological profile and molecular modeling of cyclic opioid analogues incorporating various phenylalanine derivatives.
Adamska-Bartłomiejczyk Anna, Lipiński Piotr F. J., Piekielna-Ciesielska Justyna, Kluczyk Alicja, Janecka Anna
Endomorphin-2 analogs containing modified tyrosines: Biological and theoretical investigation of the influence on conformation and pharmacological profile.
Wtorek Karol, Artali Roberto, Piekielna-Ciesielska Justyna, Koszuk Jacek, Kluczyk Alicja, Gentilucci Luca, Janecka Anna
Synthesis and pharmacological evaluation of hybrids targeting opioid and neurokinin receptors.
Wtorek Karol, Adamska-Bartłomiejczyk Anna, Piekielna-Ciesielska Justyna, Ferrari Federica, Ruzza Chiara, Kluczyk Alicja, Piasecka-Zelga Joanna, Calò Girolamo, Janecka Anna
Synthesis and activity of opioid peptidomimetics with β2- and β3-amino acids.
Gach-Janczak Katarzyna, Piekielna-Ciesielska Justyna, Adamska-Bartłomiejczyk Anna, Perlikowska Renata, Kruszyński Rafał, Kluczyk Alicja, Krzywik Julia, Sukiennik Jarosław, Cerlesi Maria Camilla, Calò Girolamo, Wasilewski Andrzej, Zielińska Marta, Janecka Anna
Synthesis, receptor binding studies, optical spectroscopic and in silico structural characterization of morphiceptin analogs with cis-4-amino-L-proline residues.
Adamska-Bartłomiejczyk Anna, Borics Attila, Tömböly Csaba, Dvorácskó Szabolcs, Lisowski Marek, Kluczyk Alicja, Wołczański Grzegorz, Piekielna-Ciesielska Justyna, Janecka Anna