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Autor publikacji Csaba Tömböly
Cyclic mu-opioid receptor ligands containing multiple N-methylated amino acid residues.
Adamska-Bartłomiejczyk Anna, Janecka Anna, Szabó Márton Richárd, Cerlesi Maria Camilla, Calò Girolamo, Kluczyk Alicja, Tömböly Csaba, Borics Attila
Synthesis, receptor binding studies, optical spectroscopic and in silico structural characterization of morphiceptin analogs with cis-4-amino-L-proline residues.
Adamska-Bartłomiejczyk Anna, Borics Attila, Tömböly Csaba, Dvorácskó Szabolcs, Lisowski Marek, Kluczyk Alicja, Wołczański Grzegorz, Piekielna-Ciesielska Justyna, Janecka Anna
Synthesis of mixed MOR/KOR efficacy cyclic opioid peptide analogs with antinociceptive activity after systemic administration.
Perlikowska Renata, Piekielna Justyna, Gentilucci Luca, De Marco Rossella, Cerlesi Maria Camilla, Calò Girolamo, Artali Roberto, Tömböly Csaba, Kluczyk Alicja, Janecka Anna
Ring size in cyclic endomorphin-2 analogs modulates receptor binding affinity and selectivity.
Piekielna Justyna, Kluczyk Alicja, Gentilucci Luca, Cerlesi Maria Camilla, Calò Girolamo, Tömböly Csaba, Łapiński Krzysztof, Janecki Tomasz, Janecka Anna
Synthesis of mixed opioid affinity cyclic endomorphin-2 analogues with fluorinated phenylalanines.
Piekielna Justyna, Perlikowska Renata, do-Rego Jean Claude, do-Rego Jean-Luc, Cerlesi Maria Camilla, Calò Girolamo, Kluczyk Alicja, Łapiński Krzysztof, Tömböly Csaba, Janecka Anna
Pharmacological characterization of endomorphin-2-based cyclic pentapeptides with methylated phenylalanine residues.
Perlikowska Renata, Malfacini Davide, Cerlesi Maria Camilla, Calò Girolamo, Piekielna Justyna, Floriot Léonore, Henry Tiphaine, do-Rego Jean Claude, Tömböly Csaba, Kluczyk Alicja, Janecka Anna