Repozytorium

Syntheses and crystal structures of three electron poor N-vinyltheophylline derivatives.

Autorzy

Ali Ramazani

A. Farshadi

Amir Tofangchi Mahyari

Katarzyna Ślepokura

Tadeusz Lis

Morteza Rouhani

Rok wydania

2011

Czasopismo

Journal of Chemical Crystallography

Numer woluminu

41

Strony

1376-1385

DOI

10.1007/s10870-011-0107-6

Kolekcja

Naukowa

Język

Angielski

Typ publikacji

Artykuł

Streszczenie

Protonation of the highly reactive 1:1 intermediates, produced in the reaction between triphenylphosphine and alkyl acetylenecarboxylates (or dialkyl acetylenedicarboxylates) by theophylline leads to vinyltriphenylphosphonium salts, which undergo Michael addition reaction with conjugate base to produce phosphorus ylides. Silica gel was found to catalyze conversion of the phosphorus ylides to electron-poor N-vinyl imidazoles in solvent-free conditions under thermal (90 °C, 1 h) conditions. The structures of these compounds were confirmed by IR, 1H, and 13C NMR spectroscopy, and single crystal X-ray structure determination. The structural analysis of the products indicated that the reaction is completely regio- and stereoselective.

Słowa kluczowe

Silica gel, Theophylline, Acetylenic esters, Vinyltriphenylphosphonium salts, crystal structure, N-Vinyl imidazole

Adres publiczny

http://dx.doi.org/10.1007/s10870-011-0107-6

Strona internetowa wydawcy

http://link.springer.com

Podobne publikacje
2008

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