Repozytorium

Iron(III) and aluminum(III) complexes with hydroxypyrone ligands aimed to design kojic acid derivatives with new perspectives.

Autorzy

Valeria Marina Nurchi

Guido Crisponi

Joanna Izabela Lachowicz

S. Murgia

T. Pivetta

Maurizio Remelli

Antonio Rescigno

Juan Niclós-Gutíerrez

Josefa M. González-Pérez

Alicia Domínguez-Martín

A. Castiñeiras

Zbigniew Szewczuk

Rok wydania

2010

Czasopismo

Journal of Inorganic Biochemistry

Numer woluminu

104

Strony

560-569

DOI

10.1016/j.jinorgbio.2010.01.007

Kolekcja

Naukowa

Język

Angielski

Typ publikacji

Artykuł

Streszczenie

With the aim to design new chelators for the clinical treatment of different diseases involving the trivalent metal ions Fe(III) and Al(III), we present the equilibria of kojic acid and its derivative 6-[5-hydroxy-2-hydroxymethyl-pyran-4-one]-5-hydroxy-2-hydroxymethyl-pyran-4-one with these two metal ions. Potentiometric and spectrophotometric techniques for iron, and potentiometry and 1H NMR for aluminum were used, supported by X-ray, electrospray ionization-mass spectrometry (ESI-MS), calorimetry and quantum chemical calculations. In this work, evidence is given on the formation of MeL, MeL2, and MeL3 complexes of both metal ions with kojic acid, confirmed by the X-ray structure of the FeL3 complex, and of variously protonated Me2L2 and MeL2 complexes of 6-[5-hydroxy-2-hydroxymethyl-pyran-4-one]-5-hydroxy-2-hydroxymethyl-pyran-4-one. The extremely good pFe value for this second ligand gives confidence to, and opens perspectives for, the search of new kojic acid derivatives.

Słowa kluczowe

Kojic acid, Fe(III), Al(III), pFe, Solution equilibria, Thermodynamic measurements, X-ray structure, molecular modeling, synthesis

Adres publiczny

https://doi.org/10.1016/j.jinorgbio.2010.01.007

Strona internetowa wydawcy

http://www.elsevier.com

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