Repozytorium
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Kolekcje
Inne
α-Amination and the 5-exo-trig cyclization reaction of sulfur-containing Schiff bases with N-phenyltriazolinedione and their anti-lipid peroxidation activity.
Autorzy
Rok wydania
2017
Czasopismo
Numer woluminu
20
Strony
424-434
DOI
10.1016/j.crci.2016.05.024
Kolekcja
Język
Angielski
Typ publikacji
Artykuł
Triazolinedione quenches efficiently the 1,2-dipoles from Schiff bases of glycine esters which are formed via a [1,2-H]-prototropic shift of their α-hydrogens, and affords the respective α-aminated products in good yields. Competition experiments show a stabilization of the 1,2-dipole from the sulfide substituent. 5-exo-trig cyclization of N-PhTAD with Schiff bases of other amino acids gave triazolines. The antioxidative and lipoxygenase inhibitory activities of the novel synthesized compounds were studied.
Słowa kluczowe
Triazolinedione, atom, amino acid, Schiff-base, α-Amination, photoluminescence
Adres publiczny
https://doi.org/10.1016/j.crci.2016.05.024
Strona internetowa wydawcy
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