Repozytorium

Amidoalkylation of phosphorus trichloride with acetamide and functionalized cyclic ketones-evidence of dominating role of side-reactions.

Autorzy

Zofia A. Dziuganowska

Iga Andrasiak

Katarzyna Ślepokura

Paweł Kafarski

Rok wydania

2014

Czasopismo

Phosphorus, Sulfur, and Silicon and the Related Elements

Numer woluminu

189

Strony

1068-1075

DOI

10.1080/10426507.2014.905573

Kolekcja

Naukowa

Język

Angielski

Typ publikacji

Artykuł

Streszczenie

The course of the reaction between phosphorus trichloride, acetamide and ethyl oxoalkanecarboxylates was studied in terms of the production of side-products. When ethyl 2-oxocycloalkane- and 4-oxocyclohexanecarboxylates were used as substrates, not only mixtures of the expected products—aminophosphonocycloalkanecarboxylic acids and their ethyl esters but also the formation of three side-products, namely 1-aminocycloalkanephosphonic acids (products of decarboxylation of the latter ones) and 1-aminoethane-1,1-diphosphonic and 1-hydroxyethane-1,1diphosphonic acids (products of the reaction of substrate and solvent with phosphonylating agent) were observed. Ethyl 2-oxo-cyclooctanecarboxylate afforded the expected 2-amino-2-pohosphonocyclooctanecarboxylic acid in minute amounts. For comparison reactions of 1-butyloxocarbonyloxopiperidines afforded the desired aminopiperidinephosphonic acids in good yields and without formation of side-products.

Słowa kluczowe

phosphonic analoques aspartic and glutamic acids, aminophosphonates, Oleksyszyn-Soroka reaction, side products

Adres publiczny

http://dx.doi.org/10.1080/10426507.2014.905573

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